Ketotifen to Boost your Clenbuterol Stack


Do you wonder how medications act in the body? How those small pieces affect your overall body systems is regulated by different receptors. The transport of each drug component through each receptor will at some point cause a degree of dysfunction with prolonged action. Thus, prolonged drug therapies affect how they are regulated in the body. So here is an example of receptor-boosting mechanism a drug does to a receptor of another.

What is Clenbuterol?

Clenbuterol is a beta-2 receptor agonist which holds function in the reversal of some degree of narrowing in the respiratory tract. Beyond its function as a bronchodilator for respiratory problems, it is one of the most preferred drugs in the facet of bodybuilding. It is classified as a thermogenic which means, it increases basal metabolic rate and core body temperature. This occurs by binding to beta-2 receptors and stimulating the mitochondria of the cells to produce and release more heat. In turn, this heats up the body’s temperature, enhances the metabolism and causes the individual to burn body fat at a greater rate. Together with an appropriate amount of exercise, proper diet, and a strong sense of self-discipline, it significantly decreases your weight and gives you a great amount of strength to enhance your performance during workout sessions. 

How does Ketotifen boost the function of Clen?

Since clenbuterol acts by binding to beta-2 receptors, this may cause a degree of down-regulation to the receptors. Like other steroids, this used to be cycled in an on and off basis because they desensitize the various receptors they act on to produce their lipolytic effect.  Ketotifen is used in conjunction with prolonged clen therapy to inhibit down-regulation of beta receptors. With the proper Ketotifen dosage for bodybuilding, it will, therefore, allow the use of these fat burning drugs for much longer periods.

Proper Administration

The best Clenbuterol and Ketotifen dosage for bodybuilding is 2 to 3 mg daily. It must be properly be administered with the right dose and duration since higher dosages may bring side effects. The dosage must also be adjusted to account for the increased effectiveness of Clen.

One disadvantage of ketotifen is that it stimulates appetite and induces hunger which counteracts the purpose of clen which is to reduce weight. A proper diet must strictly be observed to still achieve desired results.

It must be taken at night since it is an anti-histamine by nature which brings sedating effects. When taken during the day, it may cause drowsiness and may affect your circadian rhythm. Thus, giving you an abnormal sleeping pattern and may affect your strength.


As these drugs act in your body, knowing how they hold their function is a must for you to know as users. The unique function of any drug is coupled with pros and cons and being a good steward of your own body, you must need to not let the cons be greater than the pros. This article speaks about one example to manage the side effects of a drug. By this mechanism, it enhances the action of one drug and they work together with the best benefits you may get.